Patents


1. Inventor(s):
1. Abdelouahid SamadiJosé Luis Marco Contelles (Instituto de Química Orgánica General, CSIC),
2. Mercedes Unzeta, Irene Bolea (Departmento de Bioquímica; Facultat de Medicina; Universitat Autónoma de Barcelona),
3. Francisco Javier Luque (Facultat de Farmàcia, Universitat de Barcelona).
Title:        New derivatives of propargylamine having neuroprotective capacity for the treatment of Alzheimer's and Parkinson's diseases.
Date of request: 18/03/2011
International Publication number: WO/2011/113988A1
Nº of the international request: PCT/ES2011/070186
Date of the international publication: 22/09/2011
International request number: PCT/ES2011/070186
Countries: Internacional


Published in United States
Publication number: US 2013/0012522 A1
Date of publication: 10/01/2013







2.    Inventor(s): 
1. Cristóbal de los Ríos Salgado, Alejandro Romero, Javier Egea Maíquez, Rafael León, Mercedes Villarroya Sánchez, Manuela García López, Antonio García García (Universidad Autónoma de Madrid),
2. Mourad Chioua, Abdelouahid Samadi, Elena Soriano Santamaría, José Luis Marco Contelles (Instituto de Química Orgánica General, CSIC).

Title:    1,8-Naphthyridine-derived compounds and the use thereof in the treatment of neurodegenerative diseases.
Publication number: WO 2011051527 A1 20110505.
Date of publication: 2011
Countries: International


3.    Inventor(s):
1-   Abdelouahid Samadi, Mourad Chioua, Monica Alvarez Perez, Elena Soriano santamaría, Carolina Varderas y José Luis Marco Contelles, (Instituto de Química Orgánica General, CSIC),
2-   Cristobal de Los Rios, Alejandro Romero Martinez, Mercedes Villarroya Sanchez, Manuela Garcia Lopez y Antonio García García (ITH, Facultad de Medecina, UAM)

Title:    2-amino-3 ,5-dicyanopyridine and 2-chloro-3 ,5-dicyanopyridine derivatives as cholinesterase enzymes inhibitors and  with neuroprotective capacity.
Date of request: (Nº P201030377), 15/03/2010
Date of publication:27/09/2011
Publication number: ES2365233A1
Class:            Patent of invention


4.    Inventor(s): 
1.      Abdelouahid Samadi, José Luis Marco Contelles y Daniel Botelho da Silva (Instituto de Química Orgánica General de Madrid, CSIC; Juan de la Cierva, 3; 28006-Madrid).
Title:         New 2,2'-azopyridines from 2-aminopyridines of pharmaceutical and industrial interest.
Date of request: 21/06/2010
Date of publication: 18/01/2012
Publication number: ES2372342A1
Class: Patent of invention
Country: Spain


5.    Inventor(s): 
1.             Abdelouahid Samadi, José Luis Marco, David Sucunza, Mourad Chioua, (Instituto de Química Orgánica General, CSIC; Juan de la Cierva, 3; 28006-Madrid).
Title:     SÍNTESIS DE PIRIDONAS BICÍCLICAS QUE CONTIENEN EL SISTEMA HETEROCÍCLICO DE IMIDAZOL(1,2-a)PIRIDINA, A PARTIR DE 2-AMINO-6-(PROP-2-IN-1-IL AMINO) PIRIDINAS.
Date of request: 06/10/2010 (request Numbre P201031480),
Date of Publication: 19/03/2013
Publication number:          ES2379919A1
Class:            Patent of invention
Country: Spain

6. Inventor(s): 
1-    Mourad Chioua, Abdelouahid Samadi, Elena Soriano Santamaría, y José Luis Marco Contelles. (Instituto de Química Orgánica General de Madrid);
2-    Alberto Alcázar (Unidad de Proteínas, Servicio Bioquímica-Investigación,  Hospital Ramón y Cajal, Carretera de Colmenar, km 9.1, 28034-Madrid);
1-           María J. Oset-Gasque (Departamento de Bioquímica y Biología Molecular II, Facultad de Farmacia, Universidad Complutense de Madrid (UCM))
Title: QUINOLILNITRONAS
Date of request: 07.02.2013
International Publication number:  WO2013017715  (A2)
International request number: PCT/ES2012/070563
Countries: Internacional


7. Inventor(s): 
1. Mourad Chioua, Abdelouahid Samadi, Elena Soriano y José Luis Marco Contelles  (Instituto de Química Orgánica General de Madrid, CSIC).
Title:     A NEW METHOD FOR THE SYNTHESIS OF 3-methylimidazo [1,2-A] azoles: APPLICATION TO THE SYNTHESIS OF SARIPIDEM.
Date of request: (Nº P201131371),  01/08/2011
Publication number: 0617
Class:            Patent of invention
Country: Spain


8. Inventor(s): 
1-    Abdelouahid Samadi, José Luis Marco-Contelles
Consejo Superior de Investigaciones Científicas - CSIC, C/ Serrano 117, 28006 Madrid, Spain
2-    Gerard Esteban, Mercedes Unzeta
UNIVERSITAT AUTONOMA DE BARCELONA, Campus universitari s/n, 08193 Bellaterra (Cerdanyola del Valles),  Spain
3-    Li Wang, Masaki Ojima, Tsutomu Inokuchi.
National University Corporation Okayama University, 1-1, Tsushima-Naka, 1-chome, Okayama-shi, Kita-ku, Okayama 700-8530, Japan
4-    Isabel Iriepa
Universidad de Alcalá, Plaza de San Diego, s/n 28801 Alcalá de Henares, Spain.

Title: Neuroprotective multi-target directed drugs
Date of request: 30 de octubre de 2012
Publication number: EP12190483.3
Class: Patente de aplicación
Countries: European