76. E. Ramos, A.
Palomino-Antolín, M. Bartolini, I. Iriepa, I. Moraleda, D. Diez-Iriepa, A. Samadi, C. V. Cortina, M. Chioua, J.Egea,* A. Romero* and J.
Marco-Contelles*. QuinoxalineTacrine QT78, a Cholinesterase
Inhibitor as a Potential Ligand for Alzheimer’s Disease Therapy. Molecules, 24(8),1503, 2019 (IF. 3.060)
75. I. Reyes-Resina,♯ A. Samadi,*,♯ G. Navarro,♯ H. A. Saadeh,* M. A. Khasawneh,c J. Mestres, J. Marco-Contelles,* and R. Franco. Identification of a Tool Compound to Study the Mechanisms of Functional Selectivity between D 2 and D 3 Dopamine Receptors. ACS Omega, 3, 17368−17375, 2018
74. H.A. Saadeh, M.A. Khasawneh, A. Samadi,* I.A. El-Haty, G.Satała, A.J. Bojarski, L. Ismaili, Ó.M. Bautista-Aguilera, M.Yañez, J.Mestres,* and J.Marco-Contellesg,* Design, Synthesis and Biological Evaluation of Potent Antioxidant 1-(2,5-Dimethoxybenzyl)-4-arylpiperazines and N-Azolyl Substituted 2-(4-Arylpiperazin-1-yl)acetamides. ChemistrySelect, 2(13),3854-3859, 2017
75. I. Reyes-Resina,♯ A. Samadi,*,♯ G. Navarro,♯ H. A. Saadeh,* M. A. Khasawneh,c J. Mestres, J. Marco-Contelles,* and R. Franco. Identification of a Tool Compound to Study the Mechanisms of Functional Selectivity between D 2 and D 3 Dopamine Receptors. ACS Omega, 3, 17368−17375, 2018
74. H.A. Saadeh, M.A. Khasawneh, A. Samadi,* I.A. El-Haty, G.Satała, A.J. Bojarski, L. Ismaili, Ó.M. Bautista-Aguilera, M.Yañez, J.Mestres,* and J.Marco-Contellesg,* Design, Synthesis and Biological Evaluation of Potent Antioxidant 1-(2,5-Dimethoxybenzyl)-4-arylpiperazines and N-Azolyl Substituted 2-(4-Arylpiperazin-1-yl)acetamides. ChemistrySelect, 2(13),3854-3859, 2017
73. H.A. Saadeh,*
M.A. Khasawneh, Y.A. Abou-Zeid, I.A. El-Haty, S.P. Nsangou, K. Goyal, R. Sehgal, J. Marco-Contelles and A.
Samadi,* Novel 5-Nitroimidazole and 5-Nitrothiazole Peperazine Derivatives
and their Antiparasitic Activity. ChemistrySelect, 2(20), 5684–5687, 2017
72. C.Chatgilialoglu, C. Ferreri, M. Guerra, A. Samadi, and V. William Bowry. The Reaction of Thiyl Radical with Methyl Linoleate: Completing the Picture. Journal of the American Chemical Society, 139(13), 4704-4741, 2017 (IF. 14.695)
71. Marco-Contelles, J.; Serrano, M. P.; Herrero-Labrador, R.l; Romero, A.; Samadi, A.; Martínez-Murillo, R. The proof of concept of ASS234: Peripherally administered ASS234 enters the central nervous system and reduces pathology in a mouse model of Alzheimer´s disease. Journal of Psychiatry and Neuroscience: JPN, 41(1) 59-69, 2017
70 M.
Criado, J. Mulet, F. Sala, S. Sala, I. Colmena, L. Gandía, O. M.
Bautista-Aguilera, A. Samadi, M. Chioua, J. Marco-Contelles. N-benzylpiperidine derivatives
as α7 nicotinic receptor
antagonists. ACS Chemical Neuroscience, 7, 1157−1165, 2016.
69. M. Teresa Blázquez-Sánchez, F. Marcelo, M. Carmen Fernández-Alonso, R.del Villar-Guerra, A.Samadi, F. Javier Cañada, J. Jiménez-Barbero, and C. Vicent. D- and L-Mannose-containing glyco-oligoamides provide distinct recognition properties when interacting with DNA. European Journal of Organic Chemistry, 6180–6193, 2015
68. A. Samadi,* D. Da Silva, M.Chioua, L.Infantes, E. Soriano, and
J. Marco-Contelles*. The Reaction of 2-Amino-4H-pyrans with
N-Bromosuccinimide. Molecular Diversity,19, 103-122, 2015
67. O. M. Bautista-Aguilera, A. Samadi, M. Chioua, K. Nikolic, S. Filipic, D. Agbaba, E.
Soriano, S. Alcaro, R.R. Ramsay, F. Ortuso,* M. Yanez,* and J.
Marco-Contelles*.
N-Methyl-N-((1-methyl-5-(3-(1-(2-methylbenzyl)piperidin-4-yl)propoxy)-1H-indol-2-yl)methyl)prop-2-yn-1-amine,
a New Cholinesterase and Monoamine Oxidase Dual Inhibitor. Journal
of Medicinal Chemistry, 57 (24), 10455–10463, 2014
66. O. M Bautista-Aguilera, G.Esteban,
M. Chioua, K. Nikolic, D. Agbaba, I. Moraleda, I. Iriepa, E. Soriano, A. Samadi, M. Unzeta, J. Marco-Contelles. Multipotent cholinesterase/monoamine
oxidase inhibitors for the treatment of Alzheimer's disease: design, synthesis,
biochemical evaluation, ADMET, molecular modelling and QSAR analysis of novel
donepezil-pyridyl hybrids. Drug Design, Development and Therapy
2014:8, 1893–1910, 2014
65. M. Chioua, A.
Samadi, D. Postel, J. Balzarini, and J. Marco-Contelles*. Synthesis of
5-Amino-3,3-dimethyl-7-phenyl-3H-[1,2]oxathiolo[4,3-b]pyridine-6-carbonitrile
1,1-dioxides. Journal of Heterocyclic Chemistry, 51, 1452-1456, 2014
64. L.
Wang, G. Esteban, M. Ojima, O. M. Bautista-Aguilera, T. Inokuchi, I. Moraleda,
I. Iriepa, A. Samadi, M.B.H. Youdim , A. Romero, E.Soriano, R. Herrero,
A. P. Fernández Fernández, R. Martínez-Murillo, J. Marco-Contelles* and M. Unzeta. Donepezil
+ propargylamine + 8-hydroxyquinoline hybrids as new multifunctional
metal-chelators, ChE and MAO inhibitors for the potential treatment of
Alzheimer’s disease. European Journal of Medicinal Chemistry,
80, 543-561, 2014
63. Ge. Estaban, J. Allan, A. Samadi, A. Mattevi, M. Unzeta, J. Marco-Contelles, C.
Binda and R. R. Ramsay. Irreversible inhibition of human monoamine oxidases by
multi-target compounds designed for treatment of neurodegeneration. Biochimica et Biophysica Acta (BBA) - Proteins and Proteomics,
1844(6), 1104-1110, 2014
62. M. Chioua, A. Samadi, E. Soriano, L. Infantes, J. Marco-Contelles.* Silver Triflate-catalyzed Cyclization of
N2-Alkyl-N2-(prop-2-yn-1-yl)azine-2,6-diamine Derivatives leading to
1-Alkyl-3-methylene-2,3-dihydroimidazo[1,2-a]azine-5(1H)-imines**. Advanced
Synthesis & Catalysis, 356, 1235 – 1241, 2014
61. O. M. Bautista-Aguilera, G.
Esteban, I. Bolea, K. Nikolic, D. Agbaba, I. Iriepa, M. Unzeta, A. Samadi,* and J. Marco-Contelles.* Design, Synthesis, Pharmacological Evaluation, QSAR
Analysis, Molecular Modeling and ADMET of Novel Donepezil-Indolyl Hybrids as
Multipotent Cholinesterase/Monoamine Oxidase Inhibitors for the Potential
Treatment of Alzheimer’s Disease. European Journal of Medicinal Chemistry, 75, 82-95, 2014
60. María Jesús Oset-Gasque,*
María P. González, Javier Pérez-Peña, Alejandro Romero, Dimitra
Hadjipavlou-Litina, Elena Soriano, Mourad Chioua, Abdelouahid Samadi, Dushyant S. Raghuvanshi,
Krishna N. Singh,* and José Marco-Contelles*. Toxicological and Pharmacological Evaluation, Antioxidant,
ADMET and Molecular Modeling of Selected Racemic Chromenotacrines
{11-Amino-12-aryl-8,9,10,12-tetrahydro-7H-chromeno[2,3-b]quinolin-3-ols}
for the Potential Prevention and Treatment of Alzheimer’s Disease
European Journal of Medicinal Chemistry 74, 491-501, 2014
59. A. Stasiak,
M. Mussur, M. Unzeta, A. Samadi, J Marco-Contelles and W. A. Fogel.
Effects of novel monoamine oxidases and cholinesterases targeting compounds on
brain neurotransmitters and behavior in rat model of vascular dementia.
Current Pharmaceutical Design, 20(2):161-171, 2014
2013
58. I.
Bolea, A. Gella, L.Monjas, C. Pérez, M. I.Rodríguez-Franco, J. Marco-Contelles,
A. Samadi, and M. Unzeta*. Multipotent, Permeable Drug ASS234 Inhibits A-aggregation,
Possesses Antioxidant Properties and Protects SH-SY5Y Cells from A-induced
Apoptosis. Current Alzheimer Research, 10(8):797-808. 2013
57. M. Chioua, A.
Samadi, D. Postel, J. Balzarini, and J. Marco-Contelles*. Synthesis of
5-Amino-3,3-dimethyl-7-phenyl-3H-[1,2]oxathiolo[4,3-b]pyridine-6-carbonitrile
1,1-dioxides.
Journal of
Heterocyclic Chemistry,
(in press) 00,00, 2013
DOI 10.1002/jhet
DOI 10.1002/jhet
56. S. Lorrio,
A. Romero, L. González-Lafuente, R. Lajarín-Cuesta, F. J. Martínez-Sanz, M.
Estrada, A. Samadi, J. Marco-Contelles, M. Isabel Rodríguez-Franco, M.
Villarroya, M. G. López, and C.de los
Ríos*. PP2A ligand
ITH12246 protects against memory impairment and focal cerebral ischemia in
mice. ACS Chemical Neuroscience, 4(9), 1267−1277, 201355. A.
Samadi,* M. de
54. M.
Esquivias-Pérez, E. Malej, A. Romero,* F. Chabchoub, A. Samadi,
J.Marco-Contelles,* and María Jesús Oset-Gasquea.* Nontoxic and Neuroprotective β-Naphthotacrines for Alzheimer’s Disease.
Chemical Research in Toxicology, 26, 986−992, 2013
53. G.
Esteban, I. Bolea, P. Sun, M. Solé , A. Samadi, J. Marco-Contelles, and
M. Unzeta*. A therapeutic approach to cerebrovascular
diseases based on indole substituted hydrazides and hydrazines able to interact
with human Vascular Adhesion Protein-1, Monoamine Oxidases (A and B), AChE and
BuChE. Journal of Neural Transmission, 120(6):911-918,
2013
52. D. Silva, M. Chioua, A. Samadi, P. Agostinho,* P. Garcao, R. Lajarin-Cuesta, C. de los Rios, I. Iriepa, I. Moraleda, L. Gonzalez-Lafuente, M. Eduarda Mendes, C. Perez, M. Isabel Rodriguez-Franco, J. Marco-Contelles,* and M. Carmo Carreiras*. Synthesis, Pharmacological Assessment, and Molecular Modeling of Acetylcholinesterase/ButyrylcholinesteraseInhibitors: Effect against Amyloid-β-Induced Neurotoxicity. ACS Chemical Neuroscience, 4, 547−565, 2013
51. D.
Hadjipavlou-Litina*, A. Samadi, M. Unzeta, and J. Marco-Contelles*. Analysis
of the antioxidant properties of differently substituted 2- and 3-indolyl
carbohydrazides and related derivatives.
European Journal of Medicinal Chemistry, 63, 670-674, 2013
50. A. Romero,* V. Gomez-Rangel, J. Egea, A. Samadi, J. Marco-Contelles, M. G.
Lopez. Enantioselective
neuroprotective Effects of Tacripyrine ITH122 against oxygen and Glucose
Deprivation in Rat Hippocampal Slices. CNS Neuroscience & Therapeutics 19, 285–287, 2013
49. A. Romero,* R. Cacabelos, M.J. Oset-Gasque, A. Samadi, and J. Marco-Contelles,*.
Novel tacrine-related drugs as potential candidates for the treatment of
Alzheimer’s disease.
Bioorganic & Medicinal Chemistry
Letters 23, 1916–1922, 2013
48. M. Chioua, E. Soriano, L. Infantes, M. L. Jimeno,
J.Marco-Contelles and A. Samadi. The Silver-Catalyzed Cyclization of N-(Prop-2-yn-1-yl)pyridin-2-amines.
European Journal of Organic Chemistry, Volume 2013, Issue 1, 35–39, 2013
2012
47. C.Arce, S. Diaz-Castroverde, M.J. Canales, J.
Marco-Contelles, A.Samadi, M. J. Oset Gasque, and M. P. González*. Drugs for Stroke: Action of
Nitrone (Z)-N-(2-Bromo-5-hydroxy-4-methoxybenzylidene)-2-methylpropan-2-amine
oxide on Rat Cortical Neurons in Culture Subjected to
Oxygen-Glucose-Deprivation. European Journal of Medicinal Chemistry, 55, 475-479, 2012
46. A.Samadi,*
M. Estrada, C. Pérez, M.I.Rodríguez-Franco, I. Iriepa, I. Moraleda, M.Chioua,
and J. Marco-Contelles,*. Pyridonepezils; New Dual AChE inhibitors as Potential Drugs for the
Treatment of Alzheimer’s Disease: Synthesis, Biological Assessment, and
Molecular Modeling.
European Journal of Medicinal Chemistry, 57, 296-301, 2012
45. E.
Maalej, F. Chabchoub*, M. Jesús Oset-Gasque, M. Esquivias-Pérez, María P.
González, L. Monjas, C. Pérez, C. de los Ríos, M. Isabel Rodríguez-Franco, I.
Iriepa, I. Moraleda, M. Chioua, A. Romero, J. Marco-Contelles* and A. Samadi.
Synthesis, biological assessment, and
molecular modeling of racemic 7-aryl-9,10,11,12-tetrahydro-7H-benzo[7,8]chromeno[2,3-b]quinolin-8-amines
as potential drugs for the treatment of Alzheimer’s disease.
European
Journal of Medicinal Chemistry, 54, 750-763, 2012
44. A. Samadi*, C. de los
Ríos, I. Bolea, M. Chioua, I. Iriepa, I Moraleda, M. Bartolini, V. Andrisano,
E. Gálvez, C. Valderas, M. Unzeta and J. Marco-Contelles*, Multipotent MAO and
cholinesterase inhibitors for the treatment of Alzheimer’s disease: Synthesis,
pharmacological analysis and molecular modeling of heterocyclic substituted
alkyl and cycloalkyl propargyl amine.
European Journal of Medicinal Chemistry, 52,
251-262, 2012
43. M.
Chioua, D. Sucunza, E. Soriano, D. Hadjipavlou-Litina,* A. Alcazar,* I. Ayuso,
M. J. Oset-Gasque,* M. P. Gonzalez, L. Monjas, M. I. Rodriguez-Franco, J.
Marco-Contelles,* andA. Samadi. Synthesis and Antioxidant, Anti-inflammatory,
Neuroprotective and BBB Permeability. M. Chioua, D. Sucunza, E. Soriano, D. Hadjipavlou-Litina,* A. Alcázar, I.
Ayuso, M. Jesús Oset-Gasque,* M. Pilar
González, L. Monjas, M. Isabel Rodríguez-Franco, J.
Marco-Contelles,* and A. Samadi. α-Aryl-N-alkyl Nitrones, as Potential Agents for Stroke
Treatment: Synthesis, Theoretical Calculations, Antioxidant, Anti-inflammatory,
Neuroprotective, and Brain−Blood Barrier Permeability Properties. Journal of Medicinal Chemistry, 55(1), 153–168, 2012
2011
42. Stasiak,
A ; Mussur, M; Unzeta, M; Samadi, A; Marco, JL; Fogel, WA. Efects of
monoamine system directed multitarget drug on rat brain amine transmitters and
on cognitive functions in rat model of vascular dementia. Inflammation
Research, 60, Supplement: 2, S340-S341, 2011
41. I. Bolea, J.
Juárez, C. de los Ríos, M. Chioua, R. Pouplana, F. J. Luque, M. Unzeta, J.
Marco-Contelles and A. Samadi. Synthesis, Biological
Evaluation and Molecular Modelling of Donepezil and
N-[(5-(Benzyloxy)-1-methyl-1H-indol-2-yl)methyl]-N-methylprop-2-yn-1-amine
Hybrids, as New Multipotent Dual Inhibitors of Monoamine Oxidases-A/B, and
Acetyl- and Butyrylcholinesterase for the Treatment of Alzheimer’s Disease.
Journal of
Medicinal Chemistry, 54, 8251−8270, 2011
40. C. Martins, M. C. Carreiras,*
R. León, C.l de los Ríos, M. Bartolini, V. Andrisano, I. Iriepa, I. Moraleda,
E. Gálvez, M. García, J. Egea, A. Samadi,
M. Chioua, and J. Marco-Contelles*. Synthesis and biological assessment of
diversely substituted furo[2,3-b]quinolin-4-amine and pyrrolo[2,3-b]quinolin-4-amine derivatives, as novel
tacrine analogues. European Journal of Medicinal Chemistry, 46, 6119-6130, 2011
39. M.
Bartolini,* M.Pistolozzi, V. Andrisano, J. Egea, M. G. López, A.G. García, M.
Villarroya, and J. Marco-Contelles, A. Samadi. Chemical and Pharmacological Studies on
Enantiomerically Pure p-Methoxytacripyrines, Promising Multi-Target-Directed
Ligands for the Treatment of Alzheimer and Cerebrovascular Diseases. ChemMedChem, 6, 1990 –
1997, 2011
38. I.
Andreu, D. Neshchadin, E. Rico, M. Griesser, A. Samadi, I. M. Morera, G.
Gescheidt,* and M. A. Miranda*, Probing Lipid Peroxidation
by Using Linoleic Acid and Benzophenone.
Chemistry, A European Journal. 17(36), 10089-10096, 2011,
37. D. Silva, M.
Chioua, A. Samadi. M. Carmo
Carreiras, M.-L. Jimeno, E. Mendes, C. de los Ríos, A. Romero, M. Villarroya,
M. G. López, and J. Marco-Contelles, Synthesis and pharmacological assessment
of diversely substituted pyrazolo[3,4-b]quinoline, and
benzo[b]pyrazolo[4,3-g][1,8]naphthyridine derivatives. European
Journal of Medicinal Chemistry, 46,
4676-4681, 2011,
36. F.
Sánchez-Patán, M. Chioua, I. Garrido, C. Cueva, A. Samadi, J.
Marco-Contelles, M. Victoria Moreno-Arribas, B. Bartolomé, M. Monagas*.
Synthesis,
analytical features and biological relevance of 5-(3',4'-dihydroxyphenyl)--valerolactone,
a microbial metabolite derived from the catabolism of dietary flavan-3-ols. Journal
of Agricultural and Food Chemistry, 59, 7083–7091, 2011
35. J. D.
Pereira, A. Caricati-Neto, R. Miranda-Ferreira, S. Shoubi Smaili, R. O. Godinho,
C. de los Rios, R. Léon M. Villaroya,, A. Samadi, J. Marco-Contelles, N.
H. Jurkiewicz, A. G. Garcia and A. Jurkiewicz*, Effects of novel tacripyrines ITH12117 and ITH12118 on rat vas deferens
contractions, calcium transients and cholinesterase activity.
European Journal of Pharmacology, 660, 411- 419, 2011.
34. K. Mkaouar,*
F. Chabchoub,* A. Samadi, J. L.
Marco Contelles and M. Salem. A
Novel Synthesis of 14-aryl-14H-naphto[2,1-b]pyrano [3,2-e][1,2,4]triazolo[1,5-c]pyrimidins.
Heterocyclic Letters, 1(2), 96-105, 2011.
33. D. Sucunza, A. Samadi, M. Chioua,
D. B. Silva, C. Yunta, L. Infantes, M. Carmo Carreiras, E. Soriano, and J.
Marco-Contelles,*
A Practical Two-Step Synthesis of
Imidazo[1,2-a]pyridines from N-(prop-2-yn-1-yl)pyridin-2-amines.
Chemical Communications, 47,
5043–5045, 2011.
32. E. Maalej,* F. Chabchoub,* A. Samadi, C. de los Ríos, A. Perona,
A. Morreal, and J. Marco-Contelles. Synthesis, Biological
Assessment and Molecular Modelling of
14-Aryl-10,11,12,14-tetrahydro-9H-benzo[5,6]chromeno[2,3-b]quinolin-13-amines. Bioorganic
and Medicinal Chemistry Letters, 21(8), 2384-2388, 2011
31. I.Tomassoli, L. Ismaili, M. Pudlo, C. de
los Ríos, E. Soriano, I. Colmena, L. Gandía, L. Rivas, A. Samadi, J. Marco-Contelles and B. Refouvelet. Synthesis,
biological assessment and molecular modeling of new
dihydroquinoline-3-carboxamides and dihydroquinoline-3-carbohydrazide
derivatives as cholinesterase inhibitors, and Ca channel antagonists.
European Journal of
Medicinal Chemistry; 46(1), 1-10, 2011
29. A. Samadi,* D. Silva, M. Chioua, M. do Carmo
Carreiras and J.
Marco-Contelles*. Microwave
Irradiation-Assisted Amination of 2-Chloropyridine Derivatives with Amide
Solvents.
Synthetic Communications; 41, 2859-2869, 2011.
28. A.
Samadi,* E. Soriano, J. Revuelta,
C. Valderas, M. Chioua, I. Garrido,b B. Bartolomé, I. Tomassolli, L. Ismaili,
L. González-Lafuente,d M. Villarroya, A. G. García, M.J. Oset-Gasque, and . Marco-Contelles*. Synthesis, Structure, Theoretical and Experimental in
vitro Antioxidant/Pharmacological Properties of -Aryl, N-Alkyl Nitrones, as Potential
Agents for the Treatment of Cerebral Isquemia. Bioorganic and
Medicinal Chemistry; 19(2), 951–960, 2011
27. A. Samadi, C. Valderas, C. de los Ríos, A. Bastida, M.
Chioua, L. González-Lafuente, I.
Colmena, L. Gandía, A. Romero, L. del Barrio, M. D. Martín-de-Saavedra,
M. G. López,, M. Villarroya, and J.
Marco-Contelles,* Cholinergic and Neuroprotective Drugs for the Treatment of
Alzheimer and Neuronal Vascular Diseases. II. Synthesis, Biological Assessment, and Molecular
Modelling of New Tacrine Analogues from Highly Substituted
2-Aminopyridine-3-carbonitriles.
2010
26. A. Samadi, J. Marco-Contelles*, E. Soriano, M. Álvarez-Pérez, M.
Chioua, A. Romero, L. González-Lafuente, L. Gandía, J. M. Roda, M. G. López, M.
Villarroya, A.G. García, and C. de los Rios. Multipotent Drugs with Cholinergic and Neuroprotective
Properties for the Treatment of Alzheimer and Neuronal Vascular Diseases:
Synthesis, Biological Assessment, and Molecular Modelling of Simple and Readily
Available 2-Aminopyridine-, and 2-Chloropyridine-3,5-dicarbonitriles. Bioorganic
and Medicinal
Chemistry; 18, 861–5872, 2010
25. A. Stasiak, M. Unzeta, A. Samadi, J.L. Marco, W. A. Fogel. ISN'T IT HISTAMINE (HA), A UNIQUE AMINE? Conference
Information: Annual Meeting of the European-Histamine-Research-Society, JUL
13-16, 2010 Durham, ENGLAND. Inflammation Research; 59, S321-S321, 2010,
24 K. Mkaouar, F. Chabchoub, Abdelouahid Samadi, J. Louis Marco and Mansour Salem. Convenient
Synthesis of 11-aryl-1,12-dihydro-11H-naphthopyrano[2,3-d]pyrimidin-12-ones.
Synthetic
Communications; 40(22), 3405 – 3414, 2010
23. D.
Botelho da Silva, A. Samadi, L.
Infantes, M. do Carmo Carreiras and J. Marco-Contelles, Synthesis of
(E)-Diethyl 6,6'-(Diazene-1,2-diyl)bis(5-cyano-2-methyl-4-phenylnicotinates, a
New Type of 2,2’-Azopyridine Dyes. Tetrahedron.
Lett. 51, 6278–6281, 2010
22. D.
da Silva, A. Samadi,* M.Chioua, M.
do Carmo Carreiras, and J. Marco-Contellesa,* The Sandmeyer Reaction on Some
Selected Heterocyclic Ring Systems: Synthesis of Useful
2-Chloroheterocyclic-3-Carbonitrile Intermediates. Synthesis, 16,
2725–2730, 2010
21. M.
Chioua, E. Soriano, A. Samadi, and
José Marco-Contelles. Studies on
the Acetylation of 3,6-Diamino-1H-pyrazolo[3,4-b]pyridine-5-carbonitrile Derivatives.
Journal of Hyterocyclic Chemitry, 47(4), 861-872, 2010
20. C. de los Ríos, J. Egea,
J. Marco-Contelles, R. León, A. Samadi, I. González, I.Iriepa, E.
Gálvez, A. G. García, M. G. López, M. Villarroya. A. Romero. Synthesis, Inhibitory Activity of Cholinesterases and Neuroprotective
Profile of Novel 1,8-Naphthyridine Derivatives,
Journal of Medicinal Chemistry, 53(14), 5129–5143, 2010
19. E.Soriano, A. Samadi, M. Chioua, C.de los Ríos and J. Marco-Contelles, Molecular Modelling, Synthesis, and
Acetylcholinesterase Inhibition of Ethyl
5-Amino-2-methyl-6,7,8,9-tetrahydrobenzo[b][1,8]naphthyridine-3-carboxylate. Bioorg. Med. Chem. Lett., 20(9), 2950–2953, 2010
18. J.
Marco-Contelles, E. Gómez-Sánchez, A. Samadi, E. Soriano, C. Valderas,
M. Álvarez-Pérez, and M. do Carmo Carreiras. Synthesis of New
7-Azabicyclo[2.2.1]heptane Derivatives.
Arkivok;, (iii) 56-73, 2010
2009
17. M. Chioua, A. Samadi, E. Soriano, O. Lozach, L. Meijer, and J. Marco-Contelles. Synthesis and Biological Evaluation of
3,6-Diamino-1H-pyrazolo[3,4-b]pyridine Derivatives as Protein Kinase
Inhibitors. Bioorg. Med.
Chem. Lett. 19 (16),
4566-4569, 2009
16. J.
Marco-Contelles, M.ª E. Pérez-Mayoral, A.
Samadi, M.do Carmo Carreiras, and E. Soriano. Recent Advances in the Friedländer Reaction. Chemical Review. 109, 2652–2671, 2009
15. J. Marco-Contelles, R.León, C. de los Ríos, A. Samadi, M. Bartolini, V. Andrisano,
O. Huertas, X. Barril, F. Javier Luque, M. I. Rodríguez-Franco, B. López, M. G.
López, A. G. García, M. do Carmo Carreiras, and M. Villarroya. Tacripyrines, the First
Tacrine-Dihydropyridine Hybrids, as Multi-Target-Directed Ligands for the
Treatment of Alzheimer´s Disease.
Journal of Medicinal Chemistry; 52 (9), 2724-2732, 2009
14. C. Martins, A. Eleutério, M. Carmo Carreiras*,
A. Samadi, E. Soriano, R. Leon and
J. Marco-Contelles. A reinvestigation of
the acid promoted heterocyclization of 1-aryl-3,3-dicyanopropan-1-ones in the
presence of amines. Molecular Diversity; 13(4), 459–468, 2009
2001-2008
13. P.
Peñalver, A. Samadi, P. Bosch, C.
Hunter and C. Vicent. A neutral DNA sequence selective vector
for interaction studies: Fluorescence binding experiments towards a
carbohydrate-DNA carrier. Euro.
J. Org. Chem; Vol. 2008 (13), 2220–2231, 2008
12. D. Anagnostopoulos, C.
Chatgilialoglu, C. Ferreri, A. Samadi
and A. Siafaka-Kapadai. Synthesis of all-trans
arachidonic acid and its effect on rabbit platelet aggregation.
Bioorg. Med.
Chem. Lett., 15 (11): 2766-2770. 2005
11. C. Chatgilialoglu,
A. Samadi, M. Guerra, and H. Fischer. The Kinetics of Z/E Isomerization of Methyl Oleate
Catalyzed by Photogenerated Thiyl Radicals. Chem. Phys. Chem., 6(2),
286-291. 2005
10. A. Samadi, I. Andreu , C. Ferreri, S. Dellonte and C. Chatgilialoglu. Thiyl Radical Catalyzed Isomerization of Oils:
Selective Formation of Geometrical Trans Isomers.
J. Am. Oil.
Chem. Soc,
(81), 753-758, 2004
9. C. Ferreri, A. Samadi, F. Sassatelli, L. Landi, and
C. Chatgilialoglu. Regioselective Cis-Trans Isomerization of Arachidonic
Double Bonds by Thiyl Radicals: The Influence of Phospholipid Supramolecular
Organization. J. Am. Chem. Soc.; 126(4);
1063-1072, 2004
8. D. Anagnostopoulos, C. Chatgilialoglu, C.
Ferreri, A. Samadi, A. Siafaka-Kapadai. All-trans PUFA
synthesis by the thiyl radical-catalysed methodology and their effects on rabbit platelet
aggregation. Chem. Phys. Lipids., 130(1), 67, 2004
7. F. Buscá, I. Andreu , I.
M. Morera, A. Samadi and M. A.
Miranda. Chiral discrimination in the intramolecular
abstraction of allylic hydrogens by benzophenone triplets. Chem. Commun., (13),
1592 –1593, 2003
6. Ferreri C., Chatgilialoglu C., Dellonte S.,
Samadi A., Manco I. Faraone-Mennella B., Neri I., Maranini A. R. Trans-lipids formed by
a thiyl radical catalyzed process and their relevance in skin disorders. Chem. Phys.
Lipids.,
118, 90, 2002
5. M. A. Miranda, L. A
Martínez, A. Samadi, F. Buscá and I. M. Morera. Stereoselective
Intramolecular Hydrogen Abstraction by a Chiral Benzophenone Derivative.
Chemical Communications, (3), 280-281, 2002
4. A. Samadi ,
L. A. Martínez, M. A. Miranda and I. M. Morera. Mechanism of the lipid peroxidation photosensitized by
tiaprofenic acid: Product studies using linoleic acid and 1,4-cyclohexadienes
as model substrates. Photochem
and Photobiol, 73(4), 359-365, 2001
3. F. Boscá, M. A. Miranda, I. M. Morera and A.
Samadi. Involvement of type I and type II mechanisms in the linoleic acid
peroxidation photosensitized by tiaprofenic acid.
J.
Photochem and Photobiol B-Biol, 58(1), 1-5,
2000
2. R. Ballesteros, B. Abarca, A.
Samadi, J. J. Server and E. Escribá. Coordinating behaviour of
3-methyl[1,2,3]triazolo[1,5-a]pyridine (tzpy): Crystal and molecular structure
and electronic properties of [Cu(tzpy) 2 (ONO2) 2 (OH)2]. Polyhedron,18(24), 3129-3133, 1999
1.
Belén Abarca , Rafael Ballesteros, Nadia Houari and Abdelouahid Samadi. The Reaction
between Triazolobenzopyridinium and triazolothiazolium Ylides with Dimethyl
Acetylenedicarboxilate, Tetrahedron, (54), 3913-3918, 1998
